AMG-9810

AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1). Additionally, it has been shown to compete with other modes of TRPV1 activation, including proton, heat, and the endogenous ligands: anandamide, N-arachidonyl dopamine and oleoyldopamine.
Supplier Ace Therapeutics
Product # SMD097
CAS # 545395-94-6
Pricing Customizable size, Inquiry
Synonym AMG-9810; AMG9810; AMG 9810.
Product Category Lab-use Small Molecule Drugs
Chemical Formula C21H23NO3
Exact Mass 337.16779
Molecular Weight 337.41
Elemental Analysis C, 74.75; H, 6.87; N, 4.15; O, 14.23
IUPAC/Chemical Name 3-(4-t-Butylphenyl)-N-(2,3-dihydrobenzo(b)(1,4)dioxin-6-yl)acrylamide
InChi Key GZTFUVZVLYUPRG-IZZDOVSWSA-N
InChi Code InChI=1S/C21H23NO3/c1-21(2,3)16-7-4-15(5-8-16)6-11-20(23)22-17-9-10-18-19(14-17)25-13-12-24-18/h4-11,14H,12-13H2,1-3H3,(H,22,23)/b11-6+
SMILES Code CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc3c(c2)OCCO3
Appearance Solid powder
Purity >98% (or refer to the Certificate of Analysis)
Shipping Condition Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility Soluble in DMSO, not in water
Shelf Life >2 years if stored properly
Drug Formulation This drug may be formulated in DMSO
Stock Solution Storage 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code 2934.99.9001
Availability 2 Weeks
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