PHD-1-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-136300 |
| CAS # | 2009343-14-8 |
| Pricing | inquire |
| Biological Activity | PHD-1-IN-1 is an orally active and potent HIF prolylhydroxylase domain-1 (PHD-1) inhibitor with an IC50 of 0.034 μM. PHD-1-IN-1 has a unique monodentate binding interaction with the active site Fe2+ ion and induces the formation of an “Arg367-out” pocket[1]. |
| MWt | 220.23 |
| Formula | C₁₃H₈N₄ |