Imagabalin
Imagabalin, also known as PD0332334 and PF-00195889, is a drug which acts as a ligand for the α2δ subunit of the voltage-dependent calcium channel, with some selectivity for the α2δ1 subunit over α2δ2. Imagabalin has demonstrated preclinical efficacy of anxiolytic, analgesic, hypnotic, and anticonvulsant-like activity and is currently in phase III clinical trials for the treatment of generalized anxiety disorder.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD209 |
| CAS # | 610300-07-7 |
| Pricing | Customizable size, Inquiry |
| Synonym | PD 0332334; PD0332334; PD-0332334; PD 332334; PD332334; PD-332334; PF-00195889; PF 00195889; PF00195889; PF-195889; PF 195889; PF195889; Imagabalin. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C9H19NO2 |
| Exact Mass | 173.1416 |
| Molecular Weight | 173.256 |
| Elemental Analysis | C, 62.39; H, 11.05; N, 8.08; O, 18.47 |
| IUPAC/Chemical Name | (3S,5R)-3-amino-5-methyloctanoic acid |
| InChi Key | JXEHXYFSIOYTAH-SFYZADRCSA-N |
| InChi Code | InChI=1S/C9H19NO2/c1-3-4-7(2)5-8(10)6-9(11)12/h7-8H,3-6,10H2,1-2H3,(H,11,12)/t7-,8+/m1/s1 |
| SMILES Code | CCC[C@@H](C)C[C@H](N)CC(O)=O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |