BMX-IN-1
Supplier | MedChemExpress |
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Product # | HY-80002-10 mM * 1 mL |
CAS # | 1431525-23-3 |
Pricing | 10 mM * 1 mL, USD $196.0 |
Synonyms | BMX kinase inhibitor |
MWt | 524.59 |
Formula | C₂₉H₂₄N₄O₄S |
Biological Activity | BMX-IN-1 is a selective, irreversible inhibitor of bone marrow tyrosine kinase on chromosome X (BMX) that targets Cys496 in the BMX ATP binding domain with an IC50 of 8 nM, also targets the related Bruton’s tyrosine kinase (BTK) with an IC50 value of 10.4 nM, but is more than 47-656-fold less potent against Blk, JAK3, EGFR, Itk, or Tec activity. |
Purity | 99.04% |