Apelin-36(rat, mouse) TFA
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-P1065A |
| Pricing | inquire |
| Biological Activity | Apelin-36(rat, mouse) TFA is an endogenous orphan G protein-coupled receptor APJ agonist. Apelin-36(rat, mouse) TFA binds to APJ receptors with an IC50 of 5.4 nM, and potently inhibits cAMP production with an EC50 of 0.52 nM. Apelin-36(rat, mouse) TFA blocks entry of some HIV-1 and HIV-2 strains into NP-2/CD4 cells expressing APJ[1][2]. |
| MWt | 4314.91 |
| Formula | C₁₈₇H₃₀₅F₃N₆₈O₄₅S |