Desmethyl-QCA276
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-44103 |
| CAS # | 2126819-55-2 |
| Pricing | inquire |
| Biological Activity | Desmethyl-QCA276 (PROTAC BRD4-binding moiety 4), the QCA276-based moiety, binds to cereblon ligand via a linker to form PROTAC to degrade BET. QCA276 is a BET inhibitor with an IC50 of 10 nM, and with a Ki of 2.3 nM[1]. |
| Synonyms | PROTAC BRD4-binding moiety 4 |
| MWt | 387.46 |
| Formula | C₂₁H₁₇N₅OS |