PDK4-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-135954 |
| CAS # | 2310262-10-1 |
| Pricing | inquire |
| Biological Activity | PDK4-IN-1 is an anthraquinone derivative and a potent and orally active pyruvate dehydrogenase kinase 4 (PDK4) inhibitor with an IC50 value of 84 nM. PDK4-IN-1 potently represses cellular transformation and cellular proliferation and induces apoptosis. PDK4-IN-1 has antidiabetic, anticancer and anti-allergic activity[1]. |
| MWt | 357.41 |
| Formula | C₂₂H₁₉N₃O₂ |