Sarpogrelate hydrochloride

Supplier MedChemExpress
Product # HY-10564-10 mg
CAS # 135159-51-2
Pricing 10 mg, USD $75.0
Synonyms MCI-9042
MWt 465.97
Formula C₂₄H₃₂ClNO₆
Biological Activity Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, α1-, α2- and β-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis[1][2][3].
Purity ≥98.0%
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