Methiothepin mesylate
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107836-10 mM * 1 mL |
| CAS # | 74611-28-2 |
| Pricing | 10 mM * 1 mL, USD $66.0 |
| Synonyms | Metitepine mesylate; Ro 8-6837 mesylate |
| MWt | 452.65 |
| Formula | C₂₁H₂₈N₂O₃S₃ |
| Biological Activity | Methiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C). |
| Purity | ≥98.0% |