3-Bromocytisine
Supplier | MedChemExpress |
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Product # | HY-107684 |
CAS # | 207390-14-5 |
Pricing | inquire |
Biological Activity | 3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC50s are 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively[1][2]. |
Synonyms | 3-Br-cytisine |
MWt | 269.14 |
Formula | C₁₁H₁₃BrN₂O |