EGFR-IN-1 TFA
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-19617B-5 mg |
| Pricing | 5 mg, USD $480.0 |
| Biological Activity | EGFR-IN-1 TFA is an orally active and irreversible L858R/T790M mutant selective EGFR inhibitor. EGFR-IN-1 TFA potently inhibits Gefitinib-resistant EGFR L858R, T790M with 100-fold selectivity over wild-type EGFR. EGFR-IN-1 TFA displays strong antiproliferative activity against the H1975 cells and the first line mutant HCC827 cells. Antitumor activity[1]. |
| Purity | 99.05% |
| MWt | 628.6 |
| Formula | C₃₀H₃₁F₃N₆O₆ |