Zuclopenthixol acetate
Zuclopenthixol acetate is a typical antipsychotic drug of the thioxanthene class. It was introduced in 1962 by Lundbeck. Zuclopenthixol is the cis-isomer of clopenthixol. Zuclopenthixol is not approved for use in the United States. Zuclopenthixol has high affinity for both dopamine D1 and D2 receptors, for α1-adrenoceptors and 5-HT2 receptors but no affinity for cholinergic muscarine receptors. It has weak histamine (H1) receptor affinity and no α2-adrenoceptor blocking activity.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1764 |
| CAS # | 85721-05-7 (acetate) |
| Pricing | Customizable size, Inquiry |
| Synonym | Zuclopenthixol acetate; EINECS 288-415-5; UNII-349S2ZHF05 |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C24H29ClN2O2S |
| Molecular Weight | 445.02 |
| Elemental Analysis | C, 64.78; H, 6.57; Cl, 7.97; N, 6.30; O, 7.19; S, 7.20 |
| IUPAC/Chemical Name | (Z)-4-(3-(2-Chloro-9H-thioxanthen-9-ylidene)propyl)piperazine-1-ethyl acetate |
| InChi Key | DFUPOTHAXAAUMS-ZTQBIIPRSA-N |
| InChi Code | InChI=1S/C20H21ClN2S.C4H8O2/c21-15-7-8-20-18(14-15)16(17-4-1-2-6-19(17)24-20)5-3-11-23-12-9-22-10-13-23;1-3-6-4(2)5/h1-2,4-8,14,22H,3,9-13H2;3H2,1-2H3/b16-5-; |
| SMILES Code | ClC1=CC(/C2=C\CCN3CCNCC3)=C(SC4=C2C=CC=C4)C=C1.CC(OCC)=O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |