Nepicastat hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-13289A-5 mg |
| CAS # | 170151-24-3 |
| Pricing | 5 mg, USD $60.0 |
| Synonyms | SYN-117 hydrochloride; RS-25560-197 hydrochloride |
| MWt | 331.81 |
| Formula | C₁₄H₁₆ClF₂N₃S |
| Biological Activity | Nepicastat hydrochloride (SYN-117 hydrochloride) is a selective, potent, and orally active inhibitor of dopamine-beta-hydroxylase. Nepicastat hydrochloride produces concentration-dependent inhibition of bovine (IC50=8.5 nM) and human (IC50=9 nM) dopamine-beta-hydroxylase. Nepicastat hydrochloride can cross the blood-brain barrier (BBB)[1][2][3]. |
| Purity | 99.48% |