Ruboxistaurin hydrochloride

Supplier MedChemExpress
Product # HY-10195B-5 mg
CAS # 169939-93-9
Pricing 5 mg, USD $780.0
Synonyms LY333531 hydrochloride
MWt 505.01
Formula C₂₈H₂₉ClN₄O₃
Biological Activity Ruboxistaurin (LY333531) hydrochloride is an orally active, selective PKCβ inhibitor (Ki=2 nM). Ruboxistaurin hydrochloride exhibits ATP dependent competitive inhibition of PKCβI with an IC50 of 4.7 nM. Ruboxistaurin hydrochloride inhibits PKCβII with an IC50 of 5.9 nM[1][2].
Purity 99.84%
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