Ruboxistaurin hydrochloride
Supplier | MedChemExpress |
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Product # | HY-10195B-5 mg |
CAS # | 169939-93-9 |
Pricing | 5 mg, USD $780.0 |
Synonyms | LY333531 hydrochloride |
MWt | 505.01 |
Formula | C₂₈H₂₉ClN₄O₃ |
Biological Activity | Ruboxistaurin (LY333531) hydrochloride is an orally active, selective PKCβ inhibitor (Ki=2 nM). Ruboxistaurin hydrochloride exhibits ATP dependent competitive inhibition of PKCβI with an IC50 of 4.7 nM. Ruboxistaurin hydrochloride inhibits PKCβII with an IC50 of 5.9 nM[1][2]. |
Purity | 99.84% |