Agomelatine
Supplier | MedChemExpress |
---|---|
Product # | HY-17038-5 mg |
CAS # | 138112-76-2 |
Pricing | 5 mg, USD $66.0 |
Synonyms | S-20098 |
MWt | 243.3 |
Formula | C₁₅H₁₇NO₂ |
Biological Activity | Agomelatine (S-20098) is a specific agonist of MT1 and MT2 receptors with Kis of 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and HEK-hMT2, respectively[1]. Agomelatine is a selective 5-HT2C receptor antagonist with pKis of 6.4 and 6.2 at native (porcine) and cloned, human 5-HT2C receptors, respectively[2]. |
Purity | 98.77% |