Masupiridine free base
Masupiridine, also known as SUVN-502, is a 5-HT6 receptor antagonist under evulation for treating Alzheimer’s disease, attention deficit hyperactivity disorder, Parkinson’s disease and schizophrenia. SUVN-502 is a pure 5-HT6 receptor antagonist with >1200-fold selectivity over 5-HT2A receptor with a superior profile that differentiates from competitor 5-HT6 antagonists. SUVN-502 has an excellent human pharmacokinetics for once a day treatment.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1566 |
| CAS # | 701205-60-9 (free base). |
| Pricing | Customizable size, Inquiry |
| Synonym | SUVN-502; SUVN 502; SUVN502; Masupiridine; Masupiridine free base; |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C21H24BrN3O3S |
| Exact Mass | 477.0722 |
| Molecular Weight | 478.405 |
| Elemental Analysis | C, 52.72; H, 5.06; Br, 16.70; N, 8.78; O, 10.03; S, 6.70 |
| IUPAC/Chemical Name | 1-((2-bromophenyl)sulfonyl)-5-methoxy-3-((4-methylpiperazin-1-yl)methyl)-1H-indole |
| InChi Key | GWCYPEHWIZXYFZ-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C21H24BrN3O3S/c1-23-9-11-24(12-10-23)14-16-15-25(20-8-7-17(28-2)13-18(16)20)29(26,27)21-6-4-3-5-19(21)22/h3-8,13,15H,9-12,14H2,1-2H3 |
| SMILES Code | CN1CCN(CC2=CN(S(=O)(C3=CC=CC=C3Br)=O)C4=C2C=C(OC)C=C4)CC1 |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |