Ritanserin
Ritanserin (R 55667) is a selective and potent serotonin-2 antagonist. Ritanserin acts as a selective 5-HT2A (Ki = 0.45 nM) and 5-HT2C receptor (Ki = 0.71 nM) antagonist.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD361 |
| CAS # | 87051-43-2 (free base) |
| Pricing | Customizable size, Inquiry |
| Synonym | Ritanserin; R-55667; R 55667; R55667; |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C27H25F2N3OS |
| Exact Mass | 477.1686 |
| Molecular Weight | 477.57 |
| Elemental Analysis | C, 67.91; H, 5.28; F, 7.96; N, 8.80; O, 3.35; S, 6.71 |
| IUPAC/Chemical Name | 6-[2-[4-[Bis(4-fluorophenyl)methylidene]piperidin-1-yl]ethyl]-7-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one |
| InChi Key | JUQLTPCYUFPYKE-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C27H25F2N3OS/c1-18-24(26(33)32-16-17-34-27(32)30-18)12-15-31-13-10-21(11-14-31)25(19-2-6-22(28)7-3-19)20-4-8-23(29)9-5-20/h2-9,16-17H,10-15H2,1H3 |
| SMILES Code | O=C1C(CCN2CC/C(CC2)=C(C3=CC=C(F)C=C3)\C4=CC=C(F)C=C4)=C(C)N=C5N1C=CS5 |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Class-2 | Insomnia |
| Availability | 2 Weeks |