A-381393
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-116941-100 mg |
| CAS # | 726174-00-1 |
| Pricing | 100 mg, USD $950.0 |
| Biological Activity | A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM)[1]. |
| Purity | 99.96% |
| MWt | 320.43 |
| Formula | C₂₀H₂₄N₄ |