(E)-GABAB receptor antagonist 1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-129636 |
| CAS # | 1611483-29-4 |
| Pricing | inquire |
| Biological Activity | (E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist 1. GABAB receptor antagonist 1 (compound 14) is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors. (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM[1]. |
| MWt | 304.38 |
| Formula | C₁₈H₂₄O₄ |