MZ 1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107425-50 mg |
| CAS # | 1797406-69-9 |
| Pricing | 50 mg, USD $715.0 |
| Biological Activity | MZ 1 is a PROTAC BRD4 degrader. MZ 1 potently and rapidly induces reversible, long-lasting, and selective removal of BRD4 over BRD2 and BRD3. Kds of 382/120, 119/115, and 307/228 nM for BRD4 BD1/2, BRD3 BD1/2, and BRD2 BD1/2, respectively[1]. |
| Purity | ≥98.0% |
| MWt | 1002.64 |
| Formula | C₄₉H₆₀ClN₉O₈S₂ |