XMU-MP-3
XMU-MP-3 is a potent inhibitor of non-covalent BTK with IC50s of 10.7 nM and 17.0 nM for BTK WT and BTK C481S mutation in the presence of 10 μM ATP, respectively. XMU-MP-3 also induces apoptosis.
Supplier | BOC Sciences |
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Product # | 2031152-08-4 |
Pricing | Inquire |
Cas | 2031152-08-4 |
Molecular Weight | 536.55 |
Molecular Formula | C27H27F3N8O |
Canonical SMILES | CC1=C(C=C(C=C1)NC(=O)C2=CC(=CC=C2)C(F)(F)F)N3CC4=CN=C(N=C4N(C3)C)NC5=CC(=NN5C)C |