N-Desethyl Sunitinib
Supplier | MedChemExpress |
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Product # | HY-10873-10 mM * 1 mL |
CAS # | 356068-97-8 |
Pricing | 10 mM * 1 mL, USD $407.0 |
Synonyms | SU-12662 |
MWt | 370.42 |
Formula | C₂₀H₂₃FN₄O₂ |
Biological Activity | N-Desethyl Sunitinib (SU-12662) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively[1]. |
Purity | 99.35% |