N-Desethyl Sunitinib

Supplier MedChemExpress
Product # HY-10873-10 mM * 1 mL
CAS # 356068-97-8
Pricing 10 mM * 1 mL, USD $407.0
Synonyms SU-12662
MWt 370.42
Formula C₂₀H₂₃FN₄O₂
Biological Activity N-Desethyl Sunitinib (SU-12662) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively[1].
Purity 99.35%
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