S1RA hydrochloride

Supplier MedChemExpress
Product # HY-18099A-10 mM * 1 mL
CAS # 1265917-14-3
Pricing 10 mM * 1 mL, USD $121.0
Synonyms E-52862 hydrochloride
MWt 373.88
Formula C₂₀H₂₄ClN₃O₂
Biological Activity S1RA hydrochloride (E-52862 hydrochloride) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM).
Purity 99.24%
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