K-252c

Supplier MedChemExpress
Product # HY-N6736-10 mg
CAS # 85753-43-1
Pricing 10 mg, USD $460.0
Biological Activity K-252c, a staurosporine analog isolated from Nocardiopsis sp., is a cell-permeable PKC inhibitor, with an IC50 of 2.45 µM. K-252c induces apoptosis in human chronic myelogenous leukemia cancer cells. K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase[1][2][3].
MWt 311.34
Formula C₂₀H₁₃N₃O
Feedback