Zoniporide hydrochloride hydrate
Supplier | MedChemExpress |
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Product # | HY-105064D-10 mg |
CAS # | 863406-85-3 |
Pricing | 10 mg, USD $820.0 |
Synonyms | CP-597396 hydrochloride hydrate |
MWt | 374.82 |
Formula | C₁₇H₁₉ClN₆O₂ |
Biological Activity | Zoniporide (CP-597396) hydrochloride hydrate is a potent and selective inhibitor of sodium-hydrogen exchanger type 1 (NHE-1). Zoniporide hydrochloride hydrate inhibits human NHE-1 (IC50=14 nM), and has >150-fold selectivity versus other NHE isoforms. Zoniporide hydrochloride hydrate potently inhibits ex vivo NHE-1-dependent swelling of human platelets (IC50=59 nM)[1][2]. |
Purity | ≥99.0% |