GPR81 agonist 1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-135982-5 mg |
| CAS # | 1620992-67-7 |
| Pricing | 5 mg, USD $400.0 |
| Biological Activity | GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC50s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a[1]. |
| MWt | 446.63 |
| Formula | C₂₂H₃₀N₄O₂S₂ |