XE 991 dihydrochloride
Supplier | MedChemExpress |
---|---|
Product # | HY-108577-10 mM * 1 mL |
CAS # | 122955-13-9 |
Pricing | 10 mM * 1 mL, USD $165.0 |
Biological Activity | XE 991 dihydrochloride, a Kv7 (KCNQ) channels blocker, potently inhibits Kv7.1 (KCNQ1), Kv7.2 (KCNQ2), Kv7.2 + Kv7.3 (KCNQ3) channel, and M-current with IC50s of 0.75 µM, 0.71 µM, 0.6 μM, and 0.98 µM, respectively[1]. |
Purity | 98.44% |
MWt | 449.37 |
Formula | C₂₆H₂₂Cl₂N₂O |