Methotrimeprazine
Methotrimeprazine is a phenothiazine neuroleptic drug. It is a low-potency antipsychotic (approximately half as potent as chlorpromazine) with strong analgesic, hypnotic and antiemetic properties that is primarily used in palliative care. Serious side effects include tardive dyskinesia, akathisia, abnormalities in the electrical cycle of the heart, low blood pressure and the potentially fatal neuroleptic malignant syndrome. As is typical of phenothiazine antipsychotics, levomepromazine is a "dirty drug", that is, it exerts its effects by blocking a variety of receptors, including adrenergic receptors, dopamine receptors, histamine receptors, muscarinic acetylcholine receptors and serotonin receptors. (Source: https://en.wikipedia.org/wiki/Levomepromazine).
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1574 |
| CAS # | 60-99-1 |
| Pricing | Customizable size, Inquiry |
| Synonym | Levomepromazine; Nosinan; Nozinan; Levoprome. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C19H24N2OS |
| Exact Mass | 328.1609 |
| Molecular Weight | 328.474 |
| Elemental Analysis | C, 69.48; H, 7.36; N, 8.53; O, 4.87; S, 9.76 |
| IUPAC/Chemical Name | (2R)-3-(2-Methoxyphenothiazine-10-yl-)-N,N,2-trimethylpropanamine |
| InChi Key | VRQVVMDWGGWHTJ-CQSZACIVSA-N |
| InChi Code | InChI=1S/C19H24N2OS/c1-14(12-20(2)3)13-21-16-7-5-6-8-18(16)23-19-10-9-15(22-4)11-17(19)21/h5-11,14H,12-13H2,1-4H3/t14-/m1/s1 |
| SMILES Code | COC(C=C1N2C[C@H](C)CN(C)C)=CC=C1SC3=C2C=CC=C3 |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |