KDM2A/7A-IN-1
Supplier | MedChemExpress |
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Product # | HY-108706 |
CAS # | 2169272-46-0 |
Pricing | inquire |
Biological Activity | KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16 μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases[1]. |
MWt | 506.68 |
Formula | C₃₃H₃₈N₄O |