KDM2A/7A-IN-1

Supplier MedChemExpress
Product # HY-108706
CAS # 2169272-46-0
Pricing inquire
Biological Activity KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16 μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases[1].
MWt 506.68
Formula C₃₃H₃₈N₄O
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