Calmidazolium chloride
Supplier | MedChemExpress |
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Product # | HY-103319-10 mM * 1 mL |
CAS # | 57265-65-3 |
Pricing | 10 mM * 1 mL, USD $98.0 |
Synonyms | R 24571 |
MWt | 687.7 |
Formula | C₃₁H₂₃Cl₇N₂O |
Biological Activity | Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist, antagonizing CaM-dependent phosphodiesterase and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase with IC50s of 0.15 and 0.35 μM, respectively[1]. Also in anti-cancer research[2]. Calmidazolium binds to CaMK with a Kd of 3 nM. |
Purity | ≥99.0% |