ERK5-IN-2
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-128341-10 mM * 1 mL |
| CAS # | 1888305-96-1 |
| Pricing | 10 mM * 1 mL, USD $128.0 |
| Biological Activity | ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0.82 μM, 3 μM for ERK5 and ERK5 MEF2D, respectively. ERK5-IN-2 does not interact with the BRD4 bromodomain. ERK5-IN-2 suppresses both tumor xenograft growth and basic fibroblast growth factor (bFGF) driven Matrigel plug angiogenesis[1]. |
| Purity | 98.67% |
| MWt | 388.19 |
| Formula | C₁₇H₁₁BrFN₃O₂ |