Sunepitron HCl
Sunepitron, also known as CP-93,393 or CP-93,393-1 (HCl), is a combined 5-HT1A receptor agonist and α2-adrenergic receptor antagonist. It was previously under development by Pfizer for the treatment of depression and anxiety. It made it to phase III clinical trials before being discontinued.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD390 |
| CAS # | 148408-65-5 (HCl) |
| Pricing | Customizable size, Inquiry |
| Synonym | CP-93,393; CP 93,393; CP93,393; CP-93393; CP 93393; CP93393; CP-93,393-1; Sunepitron. Sunepitron HCl. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C17H24ClN5O2 |
| Molecular Weight | 365.862 |
| Elemental Analysis | C, 55.81; H, 6.61; Cl, 9.69; N, 19.14; O, 8.75 |
| IUPAC/Chemical Name | 1-(((7S,9aS)-2-(pyrimidin-2-yl)octahydro-2H-pyrido[1,2-a]pyrazin-7-yl)methyl)pyrrolidine-2,5-dione hydrochloride |
| InChi Key | HWGPYTRJVVMHGT-IODNYQNNSA-N |
| InChi Code | InChI=1S/C17H23N5O2.ClH/c23-15-4-5-16(24)22(15)11-13-2-3-14-12-21(9-8-20(14)10-13)17-18-6-1-7-19-17;/h1,6-7,13-14H,2-5,8-12H2;1H/t13-,14-;/m0./s1 |
| SMILES Code | O=C(N1C[C@H]2CC[C@@]3([H])CN(C4=NC=CC=N4)CCN3C2)CCC1=O.[H]Cl |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |