TX1-85-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100848-5 mg |
| CAS # | 1603845-32-4 |
| Pricing | 5 mg, USD $190.0 |
| Biological Activity | TX1-85-1 is an irreversible Her3 (ErbB3) inhibitor with an IC50 of 23 nM. TX1-85-1 is also the first selective Her3 ligand, which forms a covalent bond with Cys721 located in the ATP-binding site of Her3. TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling[1]. |
| Purity | ≥98.0% |
| MWt | 580.68 |
| Formula | C₃₂H₃₆N₈O₃ |