SGC-CBP30
SGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50 of 21 nM and 38 nM in cell-free assays, respectively. Exhibits 40-fold and 250-fold selectivity for CBP over the first BRD of BRD4 (BRD4(1)) and BRD4(2) respectively.
Supplier | Selleck Chemicals |
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Product # | S7256 |
Sku # | S7256-10mg |
Pricing | 10mg, $197.00 |
Citations for this product:
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bioRxiv - Systems Biology 2022Quote: ... cells were treated with 10μM SGC-CBP30 (Selleck Chemicals #S7256), 10μM tazemetostat (Selleck Chemicals #S7128) ...