GSK2656157
GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM in a cell-free assay, 500-fold greater against a panel of 300 kinases. GSK2656157 decreases apoptosis and inhibits excessive autophagy.
Supplier | Selleck Chemicals |
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Product # | S7033 |
Sku # | S7033-10mM/1mL |
Pricing | 10mM/1mL, $117.00 |
Citations for this product:
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bioRxiv - Cancer Biology 2023Quote: ... PERK inhibitor GSK2656157 (Cat#S7033) was purchased from Selleck Chemicals LLC ...