Tezampanel
Tezampanel, also known as LY 293558 and NGX-424, is a competitive antagonist of the AMPA and kainate subtypes of the ionotropic glutamate receptor family, with selectivity for the GluR5 subtype of the kainate receptor.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD404 |
| CAS # | 154652-83-2 (anhydrous) |
| Pricing | Customizable size, Inquiry |
| Synonym | LY 293558; LY-293558; LY293558; NGX-424; NGX 424; NGX424; Tezampanel |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C13H21N5O2 |
| Exact Mass | 279.1695 |
| Molecular Weight | 279.34 |
| Elemental Analysis | C, 55.90; H, 7.58; N, 25.07; O, 11.45 |
| IUPAC/Chemical Name | (3S,4aR,6R,8aR)-6-(2-(1H-tetrazol-5-yl)ethyl)decahydroisoquinoline-3-carboxylic acid |
| InChi Key | ZXFRFPSZAKNPQQ-YTWAJWBKSA-N |
| InChi Code | InChI=1S/C13H21N5O2/c19-13(20)11-6-10-5-8(1-3-9(10)7-14-11)2-4-12-15-17-18-16-12/h8-11,14H,1-7H2,(H,19,20)(H,15,16,17,18)/t8-,9+,10-,11+/m1/s1 |
| SMILES Code | O=C([C@H]1NC[C@]2([H])CC[C@H](CCC3=NN=NN3)C[C@]2([H])C1)O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | To be determined |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | To be determined |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |