Relacorilant
Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
Supplier | Selleck Chemicals |
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Product # | E1091 |
Sku # | E1091-25mg |
Pricing | 25mg, $870.00 |