CX-516

CX-516 ,aslo known as BDP 12 and SPD-420, is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator. It was researched as a treatment for Alzheimer's disease under the brand name Ampalex, and was also being examined as a treatment for ADHD. CX-516 showed good in vitro activity and positive results in animal tests, the human trials proved disappointing due mainly to low potency and short half-life. However, CX-516 is still widely used in animal research into the ampakine drugs and is the standard reference compound that newer, more potent drugs of this class such as farampator and CX-717 are compared to.
Supplier Ace Therapeutics
Product # SMD1474
CAS # 154235-83-3
Pricing Customizable size, Inquiry
Synonym CX-516; CX 516; CX516; BDP 12; BDP-12; BDP12; SPD-420; SPD420; brand name: Ampalex.
Product Category Lab-use Small Molecule Drugs
Chemical Formula C14H15N3O
Exact Mass 241.1215
Molecular Weight 241.294
Elemental Analysis C, 69.69; H, 6.27; N, 17.41; O, 6.63
IUPAC/Chemical Name 1-(quinoxalin-6-ylcarbonyl)piperidine
InChi Key ANDGGVOPIJEHOF-UHFFFAOYSA-N
InChi Code InChI=1S/C14H15N3O/c18-14(17-8-2-1-3-9-17)11-4-5-12-13(10-11)16-7-6-15-12/h4-7,10H,1-3,8-9H2
SMILES Code O=C(N1CCCCC1)C2=CC=C3N=CC=NC3=C2
Appearance Solid powder
Purity >98% (or refer to the Certificate of Analysis)
Shipping Condition Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility Soluble in DMSO, not in water
Shelf Life >2 years if stored properly
Drug Formulation This drug may be formulated in DMSO
Stock Solution Storage 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code 2934.99.9001
Availability 2 Weeks
Feedback