Glutaminase-IN-1

Supplier MedChemExpress
Product # HY-114334-50 mg
CAS # 2247127-79-1
Pricing 50 mg, USD $550.0
Synonyms CB839 derivative
MWt 618.47
Formula C₂₆H₂₄F₃N₇O₃Se
Biological Activity Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.
Purity 98.05%
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