BI-4924
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-126254-50 mg |
| CAS # | 2244452-09-1 |
| Pricing | 50 mg, USD $2650.0 |
| Biological Activity | BI-4924 is a lipophilic, highly plasma protein bound selective phosphoglycerate dehydrogenase (PHGDH) inhibitor (IC50=3 nM) with excellent microsomal, as well as hepatocytic stability. Intracellular trapping of BI-4924 disrupts serine biosynthesis with an IC50 of 2200 nM at 72 h[1]. |
| Purity | 98.48% |
| MWt | 499.36 |
| Formula | C₂₁H₂₀Cl₂N₂O₆S |