APS-2-79
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100627-5 mg |
| CAS # | 2002381-25-9 |
| Pricing | 5 mg, USD $50.0 |
| Biological Activity | APS-2-79 is a KSR-dependent MEK antagonist. APS-2-79 inhibits ATPbiotin binding to KSR2 within the KSR2-MEK1 complexe with an IC50 of 120 nM. APS-2-79 makes the stabilization of the KSR inactive state antagonizes oncogenic Ras-MAPK signaling[1]. |
| Purity | 99.31% |
| MWt | 387.43 |
| Formula | C₂₃H₂₁N₃O₃ |