AZD5153 6-hydroxy-2-naphthoic acid

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AZD5153 6-hydroxy-2-naphthoic acid (HNT salt) is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor with pKi of 8.3 for BRD4. AZD5153 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes. NSD3, via H3K36me2, acts as an epigenetic deregulator to facilitate the expression of oncogenesis-promoting genes.

Supplier	Selleck Chemicals
Product #	S8344
Sku #	S8344-25mg
Pricing	25mg, $490.00

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