KG-501 (2-naphthol-AS-E-phosphate)
KG-501 (2-naphthol-AS-E-phosphate) is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM). It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay.
Supplier | Selleck Chemicals |
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Product # | S8409 |
Sku # | S8409-10mM/1mL |
Pricing | 10mM/1mL, $99.00 |