KG-501 (2-naphthol-AS-E-phosphate)

KG-501 (2-naphthol-AS-E-phosphate) is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM). It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay.
Supplier Selleck Chemicals
Product # S8409
Sku # S8409-10mM/1mL
Pricing 10mM/1mL, $99.00
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