Desfesoterodine

Supplier MedChemExpress
Product # HY-76569-100 mg
CAS # 207679-81-0
Pricing 100 mg, USD $1488.0
Synonyms PNU-200577; 5-Hydroxymethyl Tolterodine
MWt 341.49
Formula C₂₂H₃₁NO₂
Biological Activity Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively[1]. Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053)[2][3]. Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats[4].
Purity 99.58%
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