IDH1 Inhibitor 1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-112601 |
| CAS # | 2234285-81-3 |
| Pricing | inquire |
| Biological Activity | IDH1 Inhibitor 1 is a potent, orally bioavailable, brain-penetrant and selective mutant IDH1 inhibitor with IC50s of 0.021 μM, 0.045 μM, and 2.52 μM for IDH1R132H, IDH1R132C, and IDH1WT, respectively[1]. Anticancer activity[1]. |
| MWt | 450.39 |
| Formula | C₂₀H₁₈F₄N₆O₂ |