JTV-519 free base

Supplier MedChemExpress
Product # HY-15293A
CAS # 145903-06-6
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Biological Activity JTV-519 free base (K201 free base) is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle. Antiarrhythmic and cardioprotective properties[1][2].
Synonyms K201 free base
MWt 424.6
Formula C₂₅H₃₂N₂O₂S
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