PROTAC ERα Degrader-2
Supplier | MedChemExpress |
---|---|
Product # | HY-111846-5 mg |
CAS # | 1351169-29-3 |
Pricing | 5 mg, USD $780.0 |
Biological Activity | PROTAC ERα Degrader-2 comprises a cIAP1 ligand binding group, a linker and an estrogen receptor α (ERα) binding group. PROTAC ERα Degrader-2 is an ERα degrader. Maximal ERα degradation at 30 μM concentration in human mammary tumor MCF7 cells. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs)[1]. |
Purity | 98.41% |
MWt | 763.96 |
Formula | C₄₂H₆₁N₅O₈ |