SR-4835
SR-4835 is a highly selective dual inhibitor of CDK12 and CDK13 with IC50 of 99 nM and Kd of 98 nM for CDK12 and IC50 of 4.9 nM for CDK13. SR-4835 disables triple-negative breast cancer (TNBC) cells. SR-4835 promotes synergy with DNA-damaging chemotherapy and PARP inhibitors.
Supplier | Selleck Chemicals |
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Product # | S8894 |
Sku # | S8894-10mM/1mL |
Pricing | 10mM/1mL, $459.00 |