Cyproximide
Cyproximide is a psychoactive drug discovered by American Cyanamid company. The drug exhibited activity as a central nervous system depressant and was claimed to be useful as a tranquilizing agent, hypnotic agent or muscle relaxant. The phenobarbital-like activity of cyproximide after intraperitoneal administration was demonstrated in rod traversal, clinging and righting reflex tests in mice. In addition to CNS depressant activity, cyproximide had a mild stimulant and antidepressant effects, which were shown by the restoration of exploratory behavior and an increase in locomotor activity in mice. Chronic administration of the drug led to a greater incidence of proliferative lesions in the liver of treated rats; however, the incidence of hepatocellular neoplasms was the same in treated and control rats.
Supplier | Ace Therapeutics |
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Product # | SMD780 |
CAS # | 15518-76-0 |
Pricing | Customizable size, Inquiry |
Synonym | Cyproximide; CL53415; CL-53415; CL 53415 |
Product Category | Lab-use Small Molecule Drugs |
Chemical Formula | C11H8ClNO2 |
Exact Mass | 221.0244 |
Molecular Weight | 221.64 |
Elemental Analysis | C, 59.61; H, 3.64; Cl, 15.99; N, 6.32; O, 14.44 |
IUPAC/Chemical Name | 1,2-Cyclopropanedicarboximide, 1-(p-chlorophenyl)- |
InChi Key | YYGANUVABKDFDW-UHFFFAOYSA-N |
InChi Code | InChI=1S/C11H8ClNO2/c12-7-3-1-6(2-4-7)11-5-8(11)9(14)13-10(11)15/h1-4,8H,5H2,(H,13,14,15) |
SMILES Code | O=C(C1(C2=CC=C(Cl)C=C2)C3C1)NC3=O |
Appearance | Solid powder |
Purity | >98% (or refer to the Certificate of Analysis) |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Solubility | Soluble in DMSO |
Shelf Life | >2 years if stored properly |
Drug Formulation | This drug may be formulated in DMSO |
Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
HS Tariff Code | 2934.99.9001 |