Birabresib (OTX015)
Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Supplier | Selleck Chemicals |
---|---|
Product # | S7360 |
Sku # | S7360-2mg |
Pricing | 2mg, $79.00 |